Description
of research activities
Our group`s research focuses on the molecular
and cell biology of lipid activated transcription
factors, so called nuclear receptors. Nuclear
hormone receptors are ligand activated transcription
factors participating in the regulation of cellular
proliferation, differentiation and homeostasis.
Members of this receptor superfamily, such as
the estrogen receptor, progesterone receptor or
the retinoic acid and thyroid hormone receptor
are classical endocrine regulators. According
to the general model of nuclear receptor action
in the absence of ligand receptors are bound to
corepressor complexes and transcription is inhibited.
Upon binding of agonist ligand, conformational
cahnges take place. As a consquence of these events
coregulator exchange takes place on the surface
of nuclear receptor heterodimers. After the binding
of coactivator complexes transcription of target
gene is activated.
Despite intensive studies in this field, numerous
basic questions are still need to be answered.
Our research focuses on the formation and changes
of receptor-receptor and receptor-coregulator
interactions. We apply flourescent cell imaging
techniques to address these questions. By fluorescent
correlation spectroscopy (FCS) it is possible
to investigate protein-protein interactions in
vivo, so we can study the formation and mobility
of receptor dimers and receptor-coregulator complexes
in living cells.
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